Assay Detail
Functional
CHEMBL1963983
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose response confirmation of uHTS hits that enhance the survival of human induced pluripotent stem cells when cultured as single cells in a luminescent assay. (Class of assay: confirmatory)
144
Total Activities
144
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 144 | 4.90 | 6.35 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1702179 | — | — | 1 | 6.35 |
| CHEMBL1385701 | — | — | 1 | 5.98 |
| CHEMBL1357867 | — | — | 1 | 5.96 |
| CHEMBL1865562 | — | — | 1 | 5.91 |
| CHEMBL1566415 | — | — | 1 | 5.55 |
| CHEMBL1707053 | — | — | 1 | 5.54 |
| CHEMBL510515 | — | — | 1 | 5.50 |
| CHEMBL1370276 | — | — | 1 | 5.49 |
| CHEMBL1531245 | — | — | 1 | 5.25 |
| CHEMBL1576229 | — | — | 1 | 5.23 |
| CHEMBL1990598 | — | — | 1 | 5.20 |
| CHEMBL1998338 | — | — | 1 | 5.17 |
| CHEMBL1575353 | — | — | 1 | 5.13 |
| CHEMBL338474 | HELENALIN | — | 1 | 5.10 |
| CHEMBL1319618 | — | — | 1 | 5.08 |
| CHEMBL1736090 | — | — | 1 | 5.06 |
| CHEMBL1308313 | — | — | 1 | 5.04 |
| CHEMBL1567623 | — | — | 1 | 5.03 |
| CHEMBL1728820 | — | — | 1 | 5.02 |
| CHEMBL1534791 | — | — | 1 | 5.01 |
| CHEMBL1224755 | — | — | 1 | 5.00 |
| CHEMBL1741436 | — | — | 1 | 4.97 |
| CHEMBL1906136 | — | — | 1 | 4.95 |
| CHEMBL56897 | — | — | 1 | 4.94 |
| CHEMBL1585390 | — | — | 1 | 4.89 |
| CHEMBL600694 | — | — | 1 | 4.89 |
| CHEMBL1971601 | — | — | 1 | 4.88 |
| CHEMBL1325765 | — | — | 1 | 4.87 |
| CHEMBL1597789 | — | — | 1 | 4.86 |
| CHEMBL1578828 | — | — | 1 | 4.81 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1702179 | — | EC50 | = | 448.0 | nM | 6.35 |
| CHEMBL1385701 | — | EC50 | = | 1050.0 | nM | 5.98 |
| CHEMBL1357867 | — | EC50 | = | 1110.0 | nM | 5.96 |
| CHEMBL1865562 | — | EC50 | = | 1220.0 | nM | 5.91 |
| CHEMBL1566415 | — | EC50 | = | 2810.0 | nM | 5.55 |
| CHEMBL1707053 | — | EC50 | = | 2890.0 | nM | 5.54 |
| CHEMBL510515 | — | EC50 | = | 3190.0 | nM | 5.50 |
| CHEMBL1370276 | — | EC50 | = | 3270.0 | nM | 5.49 |
| CHEMBL1531245 | — | EC50 | = | 5620.0 | nM | 5.25 |
| CHEMBL1576229 | — | EC50 | = | 5930.0 | nM | 5.23 |
| CHEMBL1990598 | — | EC50 | = | 6320.0 | nM | 5.20 |
| CHEMBL1998338 | — | EC50 | = | 6680.0 | nM | 5.17 |
| CHEMBL1575353 | — | EC50 | = | 7370.0 | nM | 5.13 |
| CHEMBL338474 | HELENALIN | EC50 | = | 7880.0 | nM | 5.10 |
| CHEMBL1319618 | — | EC50 | = | 8370.0 | nM | 5.08 |
| CHEMBL1736090 | — | EC50 | = | 8720.0 | nM | 5.06 |
| CHEMBL1308313 | — | EC50 | = | 9010.0 | nM | 5.04 |
| CHEMBL1567623 | — | EC50 | = | 9450.0 | nM | 5.03 |
| CHEMBL1728820 | — | EC50 | = | 9470.0 | nM | 5.02 |
| CHEMBL1534791 | — | EC50 | = | 9860.0 | nM | 5.01 |
| CHEMBL1224755 | — | EC50 | = | 10100.0 | nM | 5.00 |
| CHEMBL1741436 | — | EC50 | = | 10800.0 | nM | 4.97 |
| CHEMBL1906136 | — | EC50 | = | 11200.0 | nM | 4.95 |
| CHEMBL56897 | — | EC50 | = | 11500.0 | nM | 4.94 |
| CHEMBL1585390 | — | EC50 | = | 12900.0 | nM | 4.89 |
| CHEMBL600694 | — | EC50 | = | 12900.0 | nM | 4.89 |
| CHEMBL1971601 | — | EC50 | = | 13100.0 | nM | 4.88 |
| CHEMBL1325765 | — | EC50 | = | 13400.0 | nM | 4.87 |
| CHEMBL1597789 | — | EC50 | = | 13700.0 | nM | 4.86 |
| CHEMBL1537016 | — | EC50 | = | 15600.0 | nM | 4.81 |
| CHEMBL1578828 | — | EC50 | = | 15600.0 | nM | 4.81 |
| CHEMBL1534379 | — | EC50 | = | 15900.0 | nM | 4.80 |
| CHEMBL1303326 | — | EC50 | = | 20000.0 | nM | 4.70 |
| CHEMBL1890592 | — | EC50 | = | 20400.0 | nM | 4.69 |
| CHEMBL1715378 | — | EC50 | = | 20500.0 | nM | 4.69 |
| CHEMBL1554187 | — | EC50 | = | 21700.0 | nM | 4.66 |
| CHEMBL1999049 | — | EC50 | = | 24800.0 | nM | 4.61 |
| CHEMBL1304940 | — | EC50 | = | 25200.0 | nM | 4.60 |
| CHEMBL1906688 | — | EC50 | = | 25700.0 | nM | 4.59 |
| CHEMBL1563765 | — | EC50 | = | 25600.0 | nM | 4.59 |
| CHEMBL1873317 | — | EC50 | = | 26100.0 | nM | 4.58 |
| CHEMBL1361072 | — | EC50 | = | 31100.0 | nM | 4.51 |
| CHEMBL1709727 | — | EC50 | = | 30600.0 | nM | 4.51 |
| CHEMBL1346379 | — | EC50 | = | 38500.0 | nM | 4.42 |
| CHEMBL1995929 | — | EC50 | = | 37800.0 | nM | 4.42 |
| CHEMBL1964358 | — | EC50 | = | 39700.0 | nM | 4.40 |
| CHEMBL1545417 | — | EC50 | = | 41000.0 | nM | 4.39 |
| CHEMBL1598442 | — | EC50 | = | 40800.0 | nM | 4.39 |
| CHEMBL1432016 | — | EC50 | = | 42700.0 | nM | 4.37 |
| CHEMBL1414808 | — | EC50 | = | 47100.0 | nM | 4.33 |