Assay Detail
Binding
CHEMBL2013518
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Inhibition of MMP-3 using OmniMMP as substrate
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Antidotes to anthrax lethal factor intoxication. Part 3: Evaluation of core structures and further modifications to the C2-side chain.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 8 | 4.51 | 4.51 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2012838 | — | — | 1 | 4.51 |
| CHEMBL1760318 | — | — | 1 | - |
| CHEMBL2012837 | — | — | 1 | - |
| CHEMBL1760322 | — | — | 1 | - |
| CHEMBL2010824 | — | — | 1 | - |
| CHEMBL1760324 | — | — | 1 | - |
| CHEMBL2012836 | — | — | 1 | - |
| CHEMBL1269994 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2012838 | — | Ki | = | 31000.0 | nM | 4.51 |
| CHEMBL1760318 | — | Ki | > | 50000.0 | nM | - |
| CHEMBL2012837 | — | Ki | > | 50000.0 | nM | - |
| CHEMBL1760322 | — | Ki | > | 50000.0 | nM | - |
| CHEMBL2010824 | — | Ki | > | 50000.0 | nM | - |
| CHEMBL1760324 | — | Ki | > | 50000.0 | nM | - |
| CHEMBL2012836 | — | Ki | > | 50000.0 | nM | - |
| CHEMBL1269994 | — | Ki | > | 50000.0 | nM | - |