Assay Detail
Binding
CHEMBL2016156
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Inhibition of human kallikrein 1
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Human kallikrein 6 inhibitors with a para-amidobenzylanmine P1 group identified through virtual screening.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 6.80 | 7.51 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2011750 | — | — | 1 | 7.51 |
| CHEMBL2011749 | — | — | 1 | 6.09 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2011750 | — | Ki | = | 31.0 | nM | 7.51 |
| CHEMBL2011749 | — | Ki | = | 810.0 | nM | 6.09 |