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Assay Detail

CHEMBL2025706

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Hepatitis C virus genotype 1b NS5B RNA-dependent RNA polymerase P495L mutant
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Hepatitis C virus subtype 1b
Confidence 1 — Organism
Curated By Autocuration

Target

Hepatitis C virus (CHEMBL379)
Type ORGANISM
Organism Hepacivirus hominis

Publication

Hepatitis C RNA-dependent RNA polymerase inhibitors: a review of structure-activity and resistance relationships; different scaffolds and mutations.
Mayhoub AS.
Bioorg Med Chem (2012) 20 : 3150 -3161
PubMed 22516671 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.82 5.82

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL210297 1 5.82

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL210297 IC50 = 1500.0 nM 5.82