Assay Detail
Binding
CHEMBL2033709
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Inhibition of Cryptosporidium parvum CDPK1 by nonradioactive Kinaseglo luciferase assay
16
Total Activities
16
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Cryptosporidium parvum |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Multiple determinants for selective inhibition of apicomplexan calcium-dependent protein kinase CDPK1.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 16 | 8.21 | 9.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2030554 | — | — | 1 | 9.52 |
| CHEMBL2030552 | — | — | 1 | 9.40 |
| CHEMBL2030558 | — | — | 1 | 9.05 |
| CHEMBL2030553 | — | — | 1 | 8.96 |
| CHEMBL1785020 | — | — | 1 | 8.62 |
| CHEMBL2030555 | — | — | 1 | 8.62 |
| CHEMBL1241489 | — | — | 1 | 8.33 |
| CHEMBL1785021 | — | — | 1 | 8.24 |
| CHEMBL2030556 | — | — | 1 | 8.12 |
| CHEMBL1785018 | — | — | 1 | 8.10 |
| CHEMBL1242754 | — | — | 1 | 8.02 |
| CHEMBL2030561 | — | — | 1 | 7.77 |
| CHEMBL2030557 | — | — | 1 | 7.52 |
| CHEMBL2030560 | — | — | 1 | 6.55 |
| CHEMBL685 | MEBENDAZOLE | 4.0 | 1 | 6.36 |
| CHEMBL2030559 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2030554 | — | Ki | = | 0.3 | nM | 9.52 |
| CHEMBL2030552 | — | Ki | = | 0.4 | nM | 9.40 |
| CHEMBL2030558 | — | Ki | = | 0.9 | nM | 9.05 |
| CHEMBL2030553 | — | Ki | = | 1.1 | nM | 8.96 |
| CHEMBL1785020 | — | Ki | = | 2.4 | nM | 8.62 |
| CHEMBL2030555 | — | Ki | = | 2.4 | nM | 8.62 |
| CHEMBL1241489 | — | Ki | = | 4.7 | nM | 8.33 |
| CHEMBL1785021 | — | Ki | = | 5.7 | nM | 8.24 |
| CHEMBL2030556 | — | Ki | = | 7.6 | nM | 8.12 |
| CHEMBL1785018 | — | Ki | = | 8.0 | nM | 8.10 |
| CHEMBL1242754 | — | Ki | = | 9.5 | nM | 8.02 |
| CHEMBL2030561 | — | Ki | = | 17.0 | nM | 7.77 |
| CHEMBL2030557 | — | Ki | = | 30.0 | nM | 7.52 |
| CHEMBL2030560 | — | Ki | = | 280.0 | nM | 6.55 |
| CHEMBL685 | MEBENDAZOLE | Ki | = | 440.0 | nM | 6.36 |
| CHEMBL2030559 | — | Ki | > | 2500.0 | nM | - |