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Assay Detail

CHEMBL2040338

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Hepatitis C virus genotype 1b infected in human GS4.1 cells assessed as inhibition of viral replication after 72 hrs by ELISA
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Hepacivirus hominis
Confidence 1 — Organism
Curated By Autocuration

Target

Hepatitis C virus (CHEMBL379)
Type ORGANISM
Organism Hepacivirus hominis

Publication

5-acetyl-2-arylbenzimidazoles as antiviral agents. Part 4.
Vitale G, Corona P, Loriga M, Carta A, Paglietti G, Giliberti G, Sanna G, Farci P, Marongiu ME, La Colla P.
Eur J Med Chem (2012) 53 : 83 -97
PubMed 22513121 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 5.96 5.96

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2037180 1 5.96

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2037180 EC50 = 1110.0 nM 5.96