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Assay Detail

CHEMBL2044352

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antitoxoplasmic activity against Toxoplasma gondii PRU tachyzoites infected in human HFF cells assessed as beta-galactosidase activity after 72 hrs by colorimetric assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Toxoplasma gondii
Cell Type HFF
Confidence 1 — Organism
Curated By Autocuration

Target

Toxoplasma gondii (CHEMBL612888)
Type ORGANISM
Organism Toxoplasma gondii

Publication

Discovery of a new antileishmanial hit in 8-nitroquinoline series.
Paloque L, Verhaeghe P, Casanova M, Castera-Ducros C, Dumètre A, Mbatchi L, Hutter S, Kraiem-M'rabet M, Laget M, Remusat V, Rault S, Rathelot P, Azas N, Vanelle P.
Eur J Med Chem (2012) 54 : 75 -86
PubMed 22608675 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 5.18 6.10

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL36 PYRIMETHAMINE 4.0 1 6.10
CHEMBL2042573 1 4.25

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL36 PYRIMETHAMINE IC50 = 800.0 nM 6.10
CHEMBL2042573 IC50 = 56100.0 nM 4.25