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Assay Detail

CHEMBL2049534

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Functional
Antiproliferative activity against human HT-29 cells after 48 hrs by MTS assay
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HT-29
Confidence 1 — Organism
Curated By Autocuration

Target

HT-29 (CHEMBL384)
Type CELL-LINE
Organism Homo sapiens

Publication

Spectaflavoside A, a new potent iron chelating dimeric flavonol glycoside from the rhizomes of Zingiber spectabile Griff.
Sivasothy Y, Hadi AH, Mohamad K, Leong KH, Ibrahim H, Sulaiman SF, Ooi KL, Awang K.
Bioorg Med Chem Lett (2012) 22 : 3831 -3836
PubMed 22546674 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 4.82 4.95

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL378544 VINBLASTINE SULFATE 4.0 1 4.95
CHEMBL140 CURCUMIN 3.0 1 4.80
CHEMBL179512 DEMETHOXYCURCUMIN 1 4.71
CHEMBL471074 1 -
CHEMBL470049 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL378544 VINBLASTINE SULFATE IC50 = 11180.0 nM 4.95
CHEMBL140 CURCUMIN IC50 = 15900.0 nM 4.80
CHEMBL179512 DEMETHOXYCURCUMIN IC50 = 19380.0 nM 4.71
CHEMBL471074 IC50 > 150000.0 nM -
CHEMBL470049 IC50 > 150000.0 nM -