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Assay Detail

CHEMBL2061885

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiplasmodial activity against Plasmodium falciparum W2
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Plasmodium falciparum
Confidence 1 — Organism
Curated By Autocuration

Target

Plasmodium falciparum (CHEMBL364)
Type ORGANISM
Organism Plasmodium falciparum

Publication

Quinolylhydrazones as novel inhibitors of Plasmodium falciparum serine protease PfSUB1.
Gemma S, Giovani S, Brindisi M, Tripaldi P, Brogi S, Savini L, Fiorini I, Novellino E, Butini S, Campiani G, Penzo M, Blackman MJ.
Bioorg Med Chem Lett (2012) 22 : 5317 -5321
PubMed 22796182 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 6.13 6.13

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL532879 1 6.13

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL532879 EC50 = 740.0 nM 6.13