Assay Detail
Binding
CHEMBL2065347
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Inhibition of LCK
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Targeted kinase selectivity from kinase profiling data.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 7.70 | 9.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL406845 | — | — | 1 | 9.10 |
| CHEMBL1090356 | — | — | 1 | 7.40 |
| CHEMBL306380 | — | — | 1 | 7.20 |
| CHEMBL2062938 | — | — | 1 | 7.10 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL406845 | — | Ki | = | 0.7943 | nM | 9.10 |
| CHEMBL1090356 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL306380 | — | Ki | = | 63.1 | nM | 7.20 |
| CHEMBL2062938 | — | Ki | = | 79.43 | nM | 7.10 |