Assay Detail
Binding
CHEMBL2071882
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Inhibition of PDE3
35
Total Activities
35
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
Novel triazines as potent and selective phosphodiesterase 10A inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 35 | 5.71 | 6.12 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2070632 | — | — | 1 | 6.12 |
| CHEMBL2070639 | — | — | 1 | 5.91 |
| CHEMBL2070641 | — | — | 1 | 5.74 |
| CHEMBL2070671 | — | — | 1 | 5.65 |
| CHEMBL2070633 | — | — | 1 | 5.14 |
| CHEMBL2070659 | — | — | 1 | - |
| CHEMBL2069321 | — | — | 1 | - |
| CHEMBL2070658 | — | — | 1 | - |
| CHEMBL2070631 | — | — | 1 | - |
| CHEMBL2070656 | — | — | 1 | - |
| CHEMBL2070655 | — | — | 1 | - |
| CHEMBL2070654 | — | — | 1 | - |
| CHEMBL2070653 | — | — | 1 | - |
| CHEMBL2070652 | — | — | 1 | - |
| CHEMBL2070651 | — | — | 1 | - |
| CHEMBL2070650 | — | — | 1 | - |
| CHEMBL2070649 | — | — | 1 | - |
| CHEMBL2070660 | — | — | 1 | - |
| CHEMBL2070661 | — | — | 1 | - |
| CHEMBL2070662 | — | — | 1 | - |
| CHEMBL2070663 | — | — | 1 | - |
| CHEMBL2070664 | — | — | 1 | - |
| CHEMBL2070665 | — | — | 1 | - |
| CHEMBL2070666 | — | — | 1 | - |
| CHEMBL2070667 | — | — | 1 | - |
| CHEMBL2070668 | — | — | 1 | - |
| CHEMBL2070669 | — | — | 1 | - |
| CHEMBL2070670 | — | — | 1 | - |
| CHEMBL2070634 | — | — | 1 | - |
| CHEMBL2070657 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2070632 | — | IC50 | = | 750.0 | nM | 6.12 |
| CHEMBL2070639 | — | IC50 | = | 1240.0 | nM | 5.91 |
| CHEMBL2070641 | — | IC50 | = | 1820.0 | nM | 5.74 |
| CHEMBL2070671 | — | IC50 | = | 2250.0 | nM | 5.65 |
| CHEMBL2070633 | — | IC50 | = | 7260.0 | nM | 5.14 |
| CHEMBL2070631 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL2070640 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL2070656 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2070655 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2070654 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2070653 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2070652 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2070651 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2070650 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL2070649 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2069321 | — | IC50 | > | 5000.0 | nM | - |
| CHEMBL2070648 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2070647 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2070646 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2070645 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2070658 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL2070659 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL2070660 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2070661 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2070662 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2070663 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2070664 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2070665 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2070666 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2070667 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2070668 | — | IC50 | > | 5000.0 | nM | - |
| CHEMBL2070669 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2070670 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL2070634 | — | IC50 | > | 5000.0 | nM | - |
| CHEMBL2070657 | — | IC50 | > | 10000.0 | nM | - |