Assay Detail
Functional
CHEMBL2072930
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at PPARalpha
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Peroxisome proliferator-activated receptor alpha (CHEMBL239) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Targeting peroxisome proliferator-activated receptors (PPARs): development of modulators.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 5.74 | 7.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2069935 | — | — | 1 | 7.22 |
| CHEMBL565 | CLOFIBRATE | 4.0 | 1 | 4.26 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2069935 | — | EC50 | = | 60.0 | nM | 7.22 |
| CHEMBL565 | CLOFIBRATE | EC50 | = | 55000.0 | nM | 4.26 |