Assay Detail
Binding
CHEMBL2073131
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Binding affinity to Neisseria meningitidis alpha-1,4-GalT after 15 mins by competitive binding assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Neisseria meningitidis |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Inhibition of galactosyltransferases by a novel class of donor analogues.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 4.55 | 4.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL439009 | — | — | 1 | 4.77 |
| CHEMBL2070378 | — | — | 1 | 4.55 |
| CHEMBL130266 | URIDINE_DIPHOSPHATE | — | 1 | 4.34 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL439009 | — | IC50 | = | 17000.0 | nM | 4.77 |
| CHEMBL2070378 | — | IC50 | = | 28000.0 | nM | 4.55 |
| CHEMBL130266 | URIDINE_DIPHOSPHATE | IC50 | = | 46000.0 | nM | 4.34 |