Assay Detail
Functional
CHEMBL2114018
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OSM: Late stage gametocytes. IC50 values determined from 21 point dose response curves. Avery Group Griffith.
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Plasmodium falciparum NF54 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Open Source Malaria Deposition 1. http://malaria.ourexperiment.org
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 7 | 7.51 | 9.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL207990 | EPOXOMYCIN | — | 1 | 9.52 |
| CHEMBL2113939 | — | — | 1 | 8.52 |
| CHEMBL2113938 | — | — | 1 | 8.40 |
| CHEMBL2113926 | — | — | 1 | 7.55 |
| CHEMBL298470 | TAFENOQUINE | 4.0 | 1 | 5.55 |
| CHEMBL35228 | PYRONARIDINE | 3.0 | 1 | 5.53 |
| CHEMBL533269 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL207990 | EPOXOMYCIN | IC50 | = | 0.3 | nM | 9.52 |
| CHEMBL2113939 | — | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL2113938 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL2113926 | — | IC50 | = | 28.0 | nM | 7.55 |
| CHEMBL298470 | TAFENOQUINE | IC50 | = | 2800.0 | nM | 5.55 |
| CHEMBL35228 | PYRONARIDINE | IC50 | = | 2960.0 | nM | 5.53 |
| CHEMBL533269 | — | IC50 | = | - | nM | - |