Assay Detail
Binding
CHEMBL2155991
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Inhibition of LAP
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Remarkable potential of the α-aminophosphonate/phosphinate structural motif in medicinal chemistry.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 5.72 | 7.19 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2153736 | — | — | 1 | 7.19 |
| CHEMBL2153735 | — | — | 1 | 4.24 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2153736 | — | Ki | = | 65.0 | nM | 7.19 |
| CHEMBL2153735 | — | Ki | = | 58000.0 | nM | 4.24 |