Assay Detail
Binding
CHEMBL2157407
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of sodium channel site 2
2
Total Activities
1
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Discovery and development of α7 nicotinic acetylcholine receptor modulators.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 4.89 | 4.89 |
| Inhibition | 1 | - | - |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1258006 | BRADANICLINE | 2.0 | 2 | 4.89 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1258006 | BRADANICLINE | Ki | = | 13000.0 | nM | 4.89 |
| CHEMBL1258006 | BRADANICLINE | Inhibition | = | 79.0 | % | - |