Assay Detail
Functional
CHEMBL2167640
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Antagonist activity at Torpedo californica nACh receptor expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced current response
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Torpedo californica |
| Cell Type | Oocyte |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
p-(4-Azipentyl)propofol: a potent photoreactive general anesthetic derivative of propofol.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.27 | 5.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2165414 | — | — | 1 | 5.40 |
| CHEMBL526 | PROPOFOL | 4.0 | 1 | 5.14 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2165414 | — | IC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL526 | PROPOFOL | IC50 | = | 7300.0 | nM | 5.14 |