Assay Detail
Functional
CHEMBL2168752
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Agonist activity at mouse BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assay
13
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of MK-7725, A Potent, Selective Bombesin Receptor Subtype-3 Agonist for the Treatment of Obesity.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 13 | 7.02 | 7.24 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2164580 | — | — | 1 | 7.24 |
| CHEMBL2164576 | — | — | 1 | 7.24 |
| CHEMBL2164579 | — | — | 1 | 7.12 |
| CHEMBL2164223 | — | — | 1 | 7.08 |
| CHEMBL2164582 | — | — | 1 | 7.05 |
| CHEMBL2164581 | — | — | 1 | 7.03 |
| CHEMBL2164225 | — | — | 1 | 7.02 |
| CHEMBL2164226 | — | — | 1 | 7.00 |
| CHEMBL2164577 | — | — | 1 | 6.99 |
| CHEMBL2164578 | — | — | 1 | 6.94 |
| CHEMBL2023109 | — | — | 1 | 6.89 |
| CHEMBL2164222 | — | — | 1 | 6.87 |
| CHEMBL2164224 | — | — | 1 | 6.83 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2164580 | — | EC50 | = | 57.0 | nM | 7.24 |
| CHEMBL2164576 | — | EC50 | = | 58.0 | nM | 7.24 |
| CHEMBL2164579 | — | EC50 | = | 76.0 | nM | 7.12 |
| CHEMBL2164223 | — | EC50 | = | 83.0 | nM | 7.08 |
| CHEMBL2164582 | — | EC50 | = | 89.0 | nM | 7.05 |
| CHEMBL2164581 | — | EC50 | = | 93.0 | nM | 7.03 |
| CHEMBL2164225 | — | EC50 | = | 95.0 | nM | 7.02 |
| CHEMBL2164226 | — | EC50 | = | 99.0 | nM | 7.00 |
| CHEMBL2164577 | — | EC50 | = | 102.0 | nM | 6.99 |
| CHEMBL2164578 | — | EC50 | = | 115.0 | nM | 6.94 |
| CHEMBL2023109 | — | EC50 | = | 130.0 | nM | 6.89 |
| CHEMBL2164222 | — | EC50 | = | 134.0 | nM | 6.87 |
| CHEMBL2164224 | — | EC50 | = | 147.0 | nM | 6.83 |