Assay Detail
Binding
CHEMBL2168755
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [125I]-dY-peptide from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by by liquid scintillation counting
13
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of MK-7725, A Potent, Selective Bombesin Receptor Subtype-3 Agonist for the Treatment of Obesity.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 13 | 8.62 | 9.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2164581 | — | — | 1 | 9.15 |
| CHEMBL2164577 | — | — | 1 | 9.12 |
| CHEMBL2164223 | — | — | 1 | 9.05 |
| CHEMBL2164580 | — | — | 1 | 8.96 |
| CHEMBL2164582 | — | — | 1 | 8.92 |
| CHEMBL2164578 | — | — | 1 | 8.85 |
| CHEMBL2164224 | — | — | 1 | 8.77 |
| CHEMBL2164576 | — | — | 1 | 8.76 |
| CHEMBL2164222 | — | — | 1 | 8.72 |
| CHEMBL2023109 | — | — | 1 | 8.44 |
| CHEMBL2164225 | — | — | 1 | 8.08 |
| CHEMBL2164226 | — | — | 1 | 7.75 |
| CHEMBL2164579 | — | — | 1 | 7.54 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2164581 | — | IC50 | = | 0.7 | nM | 9.15 |
| CHEMBL2164577 | — | IC50 | = | 0.76 | nM | 9.12 |
| CHEMBL2164223 | — | IC50 | = | 0.9 | nM | 9.05 |
| CHEMBL2164580 | — | IC50 | = | 1.1 | nM | 8.96 |
| CHEMBL2164582 | — | IC50 | = | 1.2 | nM | 8.92 |
| CHEMBL2164578 | — | IC50 | = | 1.4 | nM | 8.85 |
| CHEMBL2164224 | — | IC50 | = | 1.7 | nM | 8.77 |
| CHEMBL2164576 | — | IC50 | = | 1.72 | nM | 8.76 |
| CHEMBL2164222 | — | IC50 | = | 1.9 | nM | 8.72 |
| CHEMBL2023109 | — | IC50 | = | 3.6 | nM | 8.44 |
| CHEMBL2164225 | — | IC50 | = | 8.3 | nM | 8.08 |
| CHEMBL2164226 | — | IC50 | = | 18.0 | nM | 7.75 |
| CHEMBL2164579 | — | IC50 | = | 29.0 | nM | 7.54 |