Assay Detail
Binding
CHEMBL2168907
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to 5-HT2C receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Structure-functional selectivity relationship studies of β-arrestin-biased dopamine D₂ receptor agonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 9.22 | 9.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2165137 | — | — | 1 | 9.22 |
| CHEMBL2165126 | — | — | 1 | 9.22 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2165137 | — | Ki | = | 0.6 | nM | 9.22 |
| CHEMBL2165126 | — | Ki | = | 0.6 | nM | 9.22 |