Assay Detail
Binding
CHEMBL2173148
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of Plasmodium falciparum MPK
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Plasmodium falciparum |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Recent results in protein kinase inhibition for tropical diseases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 5.52 | 6.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1171238 | — | — | 1 | 6.22 |
| CHEMBL1171971 | — | — | 1 | 4.82 |
| CHEMBL2171511 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1171238 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL1171971 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL2171511 | — | IC50 | = | 127000.0 | nM | - |