Assay Detail
Binding
CHEMBL2174531
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human CA2
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
The many faces of the adamantyl group in drug design.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 8.00 | 8.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1209039 | — | — | 1 | 8.10 |
| CHEMBL2170198 | — | — | 1 | 8.00 |
| CHEMBL2170197 | — | — | 1 | 7.89 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1209039 | — | Ki | = | 8.0 | nM | 8.10 |
| CHEMBL2170198 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL2170197 | — | Ki | = | 13.0 | nM | 7.89 |