Assay Detail
Binding
CHEMBL2175254
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to vasopressin V2 receptor in rabbit kidney membranes
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Oryctolagus cuniculus |
| Tissue | Kidney |
| Subcellular | Membrane |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Selective fluorescent nonpeptidic antagonists for vasopressin V₂ GPCR: application to ligand screening and oligomerization assays.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 8.13 | 8.14 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL119793 | — | — | 1 | 8.14 |
| CHEMBL603708 | — | — | 1 | 8.12 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL119793 | — | Ki | = | 7.2 | nM | 8.14 |
| CHEMBL603708 | — | Ki | = | 7.6 | nM | 8.12 |