Assay Detail
Binding
CHEMBL2184097
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Displacement of Eu-DTPA from human TLR2 expressed in HEK293 cells after 1 hr
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Novel toll-like receptor 2 ligands for targeted pancreatic cancer imaging and immunotherapy.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 7.78 | 7.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3350702 | — | — | 1 | 7.96 |
| CHEMBL2179403 | — | — | 1 | 7.60 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3350702 | — | Ki | = | 11.0 | nM | 7.96 |
| CHEMBL2179403 | — | Ki | = | 25.0 | nM | 7.60 |