Assay Detail
Binding
CHEMBL2184190
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Inhibition of Staphylococcus sp. APH(3')-3a
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Staphylococcus sp. |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
ATP-binding site of bacterial enzymes as a target for antibacterial drug design.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 5 | 4.31 | 4.31 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL143054 | — | — | 1 | 4.31 |
| CHEMBL1233654 | — | — | 1 | 4.31 |
| CHEMBL489157 | — | — | 1 | 4.31 |
| CHEMBL2181053 | — | — | 1 | 4.31 |
| CHEMBL344314 | — | — | 1 | 4.31 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL143054 | — | Ki | = | 49000.0 | nM | 4.31 |
| CHEMBL1233654 | — | Ki | = | 49000.0 | nM | 4.31 |
| CHEMBL489157 | — | Ki | = | 49000.0 | nM | 4.31 |
| CHEMBL2181053 | — | Ki | = | 49000.0 | nM | 4.31 |
| CHEMBL344314 | — | Ki | = | 49000.0 | nM | 4.31 |