Assay Detail
Functional
CHEMBL2208693
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Anti-platelet activity in human platelet-rich plasma assessed as inhibition of collagen-induced platelet aggregation
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Tissue | Plasma |
| Cell Type | Platelet |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Synopsis of some recent tactical application of bioisosteres in drug design.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 3 | 7.04 | 7.57 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL125569 | — | — | 1 | 7.57 |
| CHEMBL419780 | — | — | 1 | 6.80 |
| CHEMBL326075 | — | — | 1 | 6.75 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL125569 | — | EC50 | = | 27.0 | nM | 7.57 |
| CHEMBL419780 | — | EC50 | = | 160.0 | nM | 6.80 |
| CHEMBL326075 | — | EC50 | = | 180.0 | nM | 6.75 |