Assay Detail
Functional
CHEMBL2209156
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at human dopamine D3 receptor expressed in CHOp cells assessed as inhibition of quinpirole-induced mitogenesis after 24 hrs
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CHOp |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
CJ-1639: A Potent and Highly Selective Dopamine D3 Receptor Full Agonist.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1 | 8.77 | 8.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2203406 | — | — | 1 | 8.77 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2203406 | — | EC50 | = | 1.7 | nM | 8.77 |