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Assay Detail

CHEMBL2209399

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiproliferative activity against human U937 cells assessed as incorporation of [3H]-methyl-thymidine after 12 hrs by scintillation counting
24
Total Activities
24
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type U-937
Confidence 1 — Organism
Curated By Autocuration

Target

U-937 (CHEMBL612794)
Type CELL-LINE
Organism Homo sapiens

Publication

Structure-anti-leukemic activity relationship study of ortho-dihydroxycoumarins in U-937 cells: key role of the δ-lactone ring in determining differentiation-inducing potency and selective pro-apoptotic action.
Vázquez R, Riveiro ME, Vermeulen M, Alonso E, Mondillo C, Facorro G, Piehl L, Gómez N, Moglioni A, Fernández N, Baldi A, Shayo C, Davio C.
Bioorg Med Chem (2012) 20 : 5537 -5549
PubMed 22925447 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 24 4.05 4.08

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL276618 4-METHYLDAPHNETIN 1 4.08
CHEMBL313244 4-METHYLESCULETIN 1 4.01
CHEMBL2205242 1 -
CHEMBL458049 1 -
CHEMBL320295 O,O'-DIMETHYLCAFFEIC ACID 1 -
CHEMBL136927 DIHYDROCAFFEIC ACID 1 -
CHEMBL145 CAFFEIC ACID 3.0 1 -
CHEMBL2205241 1 -
CHEMBL54907 4-HYDROXY-6-METHYLPYRAN-2-ONE 1 -
CHEMBL372284 1 -
CHEMBL1934663 1 -
CHEMBL12626 1 -
CHEMBL6703 1 -
CHEMBL66879 COUMARIC ACID 1 -
CHEMBL1784035 1 -
CHEMBL12208 HYMECROMONE 2.0 1 -
CHEMBL2205240 1 -
CHEMBL71851 SCOPOLETIN 1 -
CHEMBL325864 SCOPARONE 1 -
CHEMBL1980149 1 -
CHEMBL12252 5,7-DIHYDROXY-4-METHYLCOUMARIN 1 -
CHEMBL244743 ESCULETIN 1 -
CHEMBL54909 FRAXETIN 1 -
CHEMBL270672 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL276618 4-METHYLDAPHNETIN IC50 = 83200.0 nM 4.08
CHEMBL313244 4-METHYLESCULETIN IC50 = 97400.0 nM 4.01
CHEMBL2205242 IC50 > 2000000.0 nM -
CHEMBL458049 IC50 > 2000000.0 nM -
CHEMBL320295 O,O'-DIMETHYLCAFFEIC ACID IC50 > 2000000.0 nM -
CHEMBL136927 DIHYDROCAFFEIC ACID IC50 = 212700.0 nM -
CHEMBL145 CAFFEIC ACID IC50 = 316500.0 nM -
CHEMBL2205241 IC50 > 2000000.0 nM -
CHEMBL54907 4-HYDROXY-6-METHYLPYRAN-2-ONE IC50 > 2000000.0 nM -
CHEMBL372284 IC50 > 2000000.0 nM -
CHEMBL1934663 IC50 > 2000000.0 nM -
CHEMBL12626 IC50 = 627700.0 nM -
CHEMBL6703 IC50 = 258700.0 nM -
CHEMBL66879 COUMARIC ACID IC50 > 2000000.0 nM -
CHEMBL1784035 IC50 = 453700.0 nM -
CHEMBL12208 HYMECROMONE IC50 = 710900.0 nM -
CHEMBL2205240 IC50 = 771300.0 nM -
CHEMBL71851 SCOPOLETIN IC50 = 975900.0 nM -
CHEMBL325864 SCOPARONE IC50 = 589900.0 nM -
CHEMBL1980149 IC50 = 736100.0 nM -
CHEMBL12252 5,7-DIHYDROXY-4-METHYLCOUMARIN IC50 > 2000000.0 nM -
CHEMBL244743 ESCULETIN IC50 = 143100.0 nM -
CHEMBL54909 FRAXETIN IC50 = 142900.0 nM -
CHEMBL270672 IC50 > 2000000.0 nM -