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Assay Detail

CHEMBL2209966

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of hemagglutininin in Influenza A virus (A/X-31(H3N2)) infected in chicken red blood cells assessed as inhibition of hemolysis preincubated for 1 hr prior to addition of red blood cells measured at pH 5.0 by spectrophotometric analysis
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Influenza A virus (A/X-31(H3N2))
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Hemagglutinin (CHEMBL4918)
Type SINGLE PROTEIN
Organism Influenza A virus (strain A/X-31 H3N2)

Publication

Microwave assisted synthesis and anti-influenza virus activity of 1-adamantyl substituted N-(1-thia-4-azaspiro[4.5]decan-4-yl)carboxamide derivatives.
Göktaş F, Vanderlinden E, Naesens L, Cesur N, Cesur Z.
Bioorg Med Chem (2012) 20 : 7155 -7159
PubMed 23117173 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 5.51 5.58

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2207987 1 5.58
CHEMBL2207978 1 5.43

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2207987 IC50 = 2600.0 nM 5.58
CHEMBL2207978 IC50 = 3700.0 nM 5.43