Assay Detail
Binding
CHEMBL2213068
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of alpha 2 adrenergic receptor by CEREP assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Optimisation of imidazole compounds as selective TAAR1 agonists: discovery of RO5073012.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 5.62 | 5.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2206397 | — | — | 1 | 5.62 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2206397 | — | Ki | = | 2400.0 | nM | 5.62 |