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Assay Detail

CHEMBL2216650

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human HeLa cells after 72 hrs by alamar blue assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HeLa
Confidence 1 — Organism
Curated By Autocuration

Target

HeLa (CHEMBL399)
Type CELL-LINE
Organism Homo sapiens

Publication

Cytotoxic cyclic depsipeptides from the Australian marine sponge Neamphius huxleyi.
Tran TD, Pham NB, Fechner G, Zencak D, Vu HT, Hooper JN, Quinn RJ.
J Nat Prod (2012) 75 : 2200 -2208
PubMed 23215348 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 6.96 7.44

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL501867 VINCRISTINE SULFATE 4.0 1 7.44
CHEMBL2208229 1 6.96
CHEMBL2208228 1 6.77
CHEMBL2208227 1 6.68

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL501867 VINCRISTINE SULFATE IC50 = 36.0 nM 7.44
CHEMBL2208229 IC50 = 110.0 nM 6.96
CHEMBL2208228 IC50 = 170.0 nM 6.77
CHEMBL2208227 IC50 = 210.0 nM 6.68