Assay Detail
Binding
CHEMBL2216694
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of para-amino phenylmercuric acetate-activated MMP2 using Mca-P-L-G-L-Dap(Dnp)-A-R-NH2 as substrate after 1 hr by fluorescence assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Design and synthesis of procollagen C-proteinase inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 4 | 6.85 | 6.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL312218 | — | — | 1 | 6.85 |
| CHEMBL2204087 | — | — | 1 | - |
| CHEMBL2204807 | — | — | 1 | - |
| CHEMBL2204802 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL312218 | — | IC50 | = | 140.0 | nM | 6.85 |
| CHEMBL2204087 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL2204807 | — | IC50 | > | 6000.0 | nM | - |
| CHEMBL2204802 | — | IC50 | > | 25000.0 | nM | - |