Assay Detail
Binding
CHEMBL2217067
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Competitive inhibition of carnitine palmitoyltransferase using palmitoyl-CoA
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Carnitine palmitoyltransferase (CPT) modulators: a medicinal chemistry perspective on 35 years of research.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 6.16 | 6.60 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL307495 | — | — | 1 | 6.60 |
| CHEMBL1231506 | TEGLICAR | 2.0 | 1 | 6.44 |
| CHEMBL114113 | — | — | 1 | 5.44 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL307495 | — | Ki | = | 250.0 | nM | 6.60 |
| CHEMBL1231506 | TEGLICAR | Ki | = | 360.0 | nM | 6.44 |
| CHEMBL114113 | — | Ki | = | 3600.0 | nM | 5.44 |