Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL2217256

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of JNK2
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Mitogen-activated protein kinase 9 (CHEMBL4179)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Irreversible protein kinase inhibitors: balancing the benefits and risks.
Barf T, Kaptein A.
J Med Chem (2012) 55 : 6243 -6262
PubMed 22621397 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.73 7.73

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2216824 1 7.73

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2216824 IC50 = 18.7 nM 7.73