Assay Detail
Binding
CHEMBL2321339
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Inhibition of IL-5 in mouse pro-B Y16 cells after 48 hrs by WST1 assay
28
Total Activities
28
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Cell Type | Y16 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Identification of novel chromenone derivatives as interleukin-5 inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 28 | 4.91 | 5.24 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1164199 | — | — | 1 | 5.24 |
| CHEMBL2316354 | — | — | 1 | 5.19 |
| CHEMBL2316357 | — | — | 1 | 5.17 |
| CHEMBL2316356 | — | — | 1 | 5.16 |
| CHEMBL2316353 | — | — | 1 | 5.16 |
| CHEMBL486626 | SOPHORICOSIDE | — | 1 | 4.97 |
| CHEMBL2316358 | — | — | 1 | 4.90 |
| CHEMBL2316373 | — | — | 1 | 4.90 |
| CHEMBL2316355 | — | — | 1 | 4.88 |
| CHEMBL2316351 | — | — | 1 | 4.82 |
| CHEMBL2316374 | — | — | 1 | 4.82 |
| CHEMBL2316375 | — | — | 1 | 4.80 |
| CHEMBL2316361 | — | — | 1 | 4.79 |
| CHEMBL2316365 | — | — | 1 | 4.74 |
| CHEMBL2316360 | — | — | 1 | 4.72 |
| CHEMBL2316364 | — | — | 1 | 4.60 |
| CHEMBL1370 | BUDESONIDE | 4.0 | 1 | 4.57 |
| CHEMBL2316362 | — | — | 1 | - |
| CHEMBL2316363 | — | — | 1 | - |
| CHEMBL2316359 | — | — | 1 | - |
| CHEMBL2316366 | — | — | 1 | - |
| CHEMBL2316367 | — | — | 1 | - |
| CHEMBL2316368 | — | — | 1 | - |
| CHEMBL2316369 | — | — | 1 | - |
| CHEMBL2316370 | — | — | 1 | - |
| CHEMBL2316371 | — | — | 1 | - |
| CHEMBL2316372 | — | — | 1 | - |
| CHEMBL2316352 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1164199 | — | IC50 | = | 5800.0 | nM | 5.24 |
| CHEMBL2316354 | — | IC50 | = | 6400.0 | nM | 5.19 |
| CHEMBL2316357 | — | IC50 | = | 6700.0 | nM | 5.17 |
| CHEMBL2316356 | — | IC50 | = | 7000.0 | nM | 5.16 |
| CHEMBL2316353 | — | IC50 | = | 7000.0 | nM | 5.16 |
| CHEMBL486626 | SOPHORICOSIDE | IC50 | = | 10600.0 | nM | 4.97 |
| CHEMBL2316358 | — | IC50 | = | 12600.0 | nM | 4.90 |
| CHEMBL2316373 | — | IC50 | = | 12500.0 | nM | 4.90 |
| CHEMBL2316355 | — | IC50 | = | 13200.0 | nM | 4.88 |
| CHEMBL2316351 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL2316374 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL2316375 | — | IC50 | = | 16000.0 | nM | 4.80 |
| CHEMBL2316361 | — | IC50 | = | 16200.0 | nM | 4.79 |
| CHEMBL2316365 | — | IC50 | = | 18100.0 | nM | 4.74 |
| CHEMBL2316360 | — | IC50 | = | 19100.0 | nM | 4.72 |
| CHEMBL2316364 | — | IC50 | = | 25100.0 | nM | 4.60 |
| CHEMBL1370 | BUDESONIDE | IC50 | = | 27100.0 | nM | 4.57 |
| CHEMBL2316362 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL2316363 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL2316359 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL2316366 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL2316367 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL2316368 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL2316369 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL2316370 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL2316371 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL2316372 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL2316352 | — | IC50 | > | 30000.0 | nM | - |