Assay Detail
Binding
CHEMBL2327422
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Positive modulatory activity at voltage-gated K channel 7.5 (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Potassium voltage-gated channel subfamily KQT member 5 (CHEMBL2925) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Ion channels as therapeutic targets: a drug discovery perspective.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1 | 5.62 | 5.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL266510 | FLINDOKALNER | 3.0 | 1 | 5.62 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL266510 | FLINDOKALNER | EC50 | = | 2400.0 | nM | 5.62 |