Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL2328927

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of UBA7 (unknown origin) in presence of ATP
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Ubiquitin-like modifier-activating enzyme 7 (CHEMBL2321623)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Exploring a new frontier in cancer treatment: targeting the ubiquitin and ubiquitin-like activating enzymes.
da Silva SR, Paiva SL, Lukkarila JL, Gunning PT.
J Med Chem (2013) 56 : 2165 -2177
PubMed 23360215 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.40 5.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2017005 1 5.40

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2017005 IC50 = 4000.0 nM 5.40