Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL2330482

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiparasitic activity against tachyzoites of Toxoplasma gondii RH type 1 infected in HFF cells incubated for 4 hrs followed by compound washout measured after 72 hrs by beta-galactoside reporter assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Toxoplasma gondii
Cell Type HFF
Confidence 1 — Organism
Curated By Autocuration

Target

Toxoplasma gondii (CHEMBL612888)
Type ORGANISM
Organism Toxoplasma gondii

Publication

Optimizing small molecule inhibitors of calcium-dependent protein kinase 1 to prevent infection by Toxoplasma gondii.
Lourido S, Zhang C, Lopez MS, Tang K, Barks J, Wang Q, Wildman SA, Shokat KM, Sibley LD.
J Med Chem (2013) 56 : 3068 -3077
PubMed 23470217 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 7.00 7.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1236661 1 7.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1236661 EC50 = 100.0 nM 7.00