Assay Detail
Binding
CHEMBL2339941
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of Staphylococcus aureus AgrC4
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Staphylococcus aureus |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Attenuating Staphylococcus aureus virulence gene regulation: a medicinal chemistry perspective.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 4 | 7.26 | 8.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2337555 | — | — | 1 | 8.52 |
| CHEMBL2337558 | — | — | 1 | 8.30 |
| CHEMBL1823954 | — | — | 1 | 6.82 |
| CHEMBL2337557 | — | — | 1 | 5.39 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2337555 | — | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL2337558 | — | IC50 | = | 5.0 | nM | 8.30 |
| CHEMBL1823954 | — | IC50 | = | 150.0 | nM | 6.82 |
| CHEMBL2337557 | — | IC50 | = | 4100.0 | nM | 5.39 |