Assay Detail
Binding
CHEMBL2341185
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Inhibition of human recombinant ARTD1 by fluorescence assay
18
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Screening and structural analysis of flavones inhibiting tankyrases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 18 | 5.23 | 5.90 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL222556 | — | — | 2 | 5.90 |
| CHEMBL275638 | FLAVONE | 2.0 | 2 | 5.86 |
| CHEMBL147552 | — | — | 2 | 5.62 |
| CHEMBL151 | LUTEOLIN | 2.0 | 2 | 5.38 |
| CHEMBL301624 | — | — | 2 | 5.12 |
| CHEMBL253786 | — | — | 2 | 5.02 |
| CHEMBL53738 | — | — | 2 | 5.00 |
| CHEMBL16861 | — | — | 2 | 4.60 |
| CHEMBL28 | APIGENIN | — | 1 | 4.00 |
| CHEMBL16751 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL222556 | — | IC50 | = | 1258.93 | nM | 5.90 |
| CHEMBL222556 | — | IC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL275638 | FLAVONE | IC50 | = | 1380.38 | nM | 5.86 |
| CHEMBL275638 | FLAVONE | IC50 | = | 1400.0 | nM | 5.85 |
| CHEMBL147552 | — | IC50 | = | 2400.0 | nM | 5.62 |
| CHEMBL147552 | — | IC50 | = | 2454.71 | nM | 5.61 |
| CHEMBL151 | LUTEOLIN | IC50 | = | 4200.0 | nM | 5.38 |
| CHEMBL151 | LUTEOLIN | IC50 | = | 4265.8 | nM | 5.37 |
| CHEMBL301624 | — | IC50 | = | 7585.78 | nM | 5.12 |
| CHEMBL301624 | — | IC50 | = | 7500.0 | nM | 5.12 |
| CHEMBL253786 | — | IC50 | = | 9549.93 | nM | 5.02 |
| CHEMBL253786 | — | IC50 | = | 9500.0 | nM | 5.02 |
| CHEMBL53738 | — | IC50 | = | 9900.0 | nM | 5.00 |
| CHEMBL53738 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL16861 | — | IC50 | = | 25000.0 | nM | 4.60 |
| CHEMBL16861 | — | IC50 | = | 25703.96 | nM | 4.59 |
| CHEMBL28 | APIGENIN | IC50 | = | 100000.0 | nM | 4.00 |
| CHEMBL16751 | — | IC50 | > | 100000.0 | nM | - |