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Assay Detail

CHEMBL2342808

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antimalarial activity against chloroquine-resistant Plasmodium falciparum ItG after 72 hrs by lactate dehydrogenase assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Plasmodium falciparum
Confidence 1 — Organism
Curated By Autocuration

Target

Plasmodium falciparum (CHEMBL364)
Type ORGANISM
Organism Plasmodium falciparum

Publication

Antimalarial activities of 6-iodouridine and its prodrugs and potential for combination therapy.
Crandall IE, Wasilewski E, Bello AM, Mohmmed A, Malhotra P, Pai EF, Kain KC, Kotra LP.
J Med Chem (2013) 56 : 2348 -2358
PubMed 23410043 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 6.31 6.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL76 CHLOROQUINE 4.0 1 6.70
CHEMBL220442 1 5.92

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL76 CHLOROQUINE IC50 = 200.0 nM 6.70
CHEMBL220442 IC50 = 1200.0 nM 5.92