Assay Detail
Functional
CHEMBL2354232
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PubChem BioAssay. Counterscreen for antagonists of the human trace amine associated receptor 1 (hTAAR1): Fluorescence-based cell-based high throughput dose response assay to identify nonselective Ga16 antagonists. (Class of assay: confirmatory)
40
Total Activities
40
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 40 | 4.74 | 5.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1599142 | — | — | 1 | 5.00 |
| CHEMBL1481854 | — | — | 1 | 4.87 |
| CHEMBL3209047 | — | — | 1 | 4.82 |
| CHEMBL1710088 | — | — | 1 | 4.76 |
| CHEMBL3199120 | — | — | 1 | 4.55 |
| CHEMBL1603221 | — | — | 1 | 4.42 |
| CHEMBL1603300 | — | — | 1 | - |
| CHEMBL1482973 | — | — | 1 | - |
| CHEMBL1564914 | — | — | 1 | - |
| CHEMBL1375903 | — | — | 1 | - |
| CHEMBL1521368 | — | — | 1 | - |
| CHEMBL1704306 | — | — | 1 | - |
| CHEMBL1386399 | — | — | 1 | - |
| CHEMBL1404043 | — | — | 1 | - |
| CHEMBL2355870 | — | — | 1 | - |
| CHEMBL3198435 | — | — | 1 | - |
| CHEMBL1700821 | — | — | 1 | - |
| CHEMBL3196777 | — | — | 1 | - |
| CHEMBL1999268 | — | — | 1 | - |
| CHEMBL3190072 | — | — | 1 | - |
| CHEMBL1402878 | — | — | 1 | - |
| CHEMBL3189778 | — | — | 1 | - |
| CHEMBL1315467 | — | — | 1 | - |
| CHEMBL1476854 | — | — | 1 | - |
| CHEMBL3191107 | — | — | 1 | - |
| CHEMBL1593829 | — | — | 1 | - |
| CHEMBL3208641 | — | — | 1 | - |
| CHEMBL1362116 | — | — | 1 | - |
| CHEMBL1877432 | — | — | 1 | - |
| CHEMBL1525419 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1599142 | — | IC50 | = | 10023.0 | nM | 5.00 |
| CHEMBL1481854 | — | IC50 | = | 13478.0 | nM | 4.87 |
| CHEMBL3209047 | — | IC50 | = | 15278.0 | nM | 4.82 |
| CHEMBL1710088 | — | IC50 | = | 17494.0 | nM | 4.76 |
| CHEMBL3199120 | — | IC50 | = | 28070.0 | nM | 4.55 |
| CHEMBL1603221 | — | IC50 | = | 38351.0 | nM | 4.42 |
| CHEMBL1386399 | — | IC50 | > | 29916.0 | nM | - |
| CHEMBL1336531 | — | IC50 | > | 29913.0 | nM | - |
| CHEMBL1404043 | — | IC50 | > | 29906.0 | nM | - |
| CHEMBL2355870 | — | IC50 | > | 29881.0 | nM | - |
| CHEMBL3198435 | — | IC50 | > | 29910.0 | nM | - |
| CHEMBL1700821 | — | IC50 | > | 29900.0 | nM | - |
| CHEMBL3196777 | — | IC50 | > | 29934.0 | nM | - |
| CHEMBL1482973 | — | IC50 | > | 29910.0 | nM | - |
| CHEMBL1427061 | — | IC50 | > | 29909.0 | nM | - |
| CHEMBL1531065 | — | IC50 | > | 29919.0 | nM | - |
| CHEMBL1561828 | — | IC50 | > | 29909.0 | nM | - |
| CHEMBL1372064 | — | IC50 | > | 29910.0 | nM | - |
| CHEMBL1318522 | — | IC50 | > | 29884.0 | nM | - |
| CHEMBL1451260 | — | IC50 | > | 29913.0 | nM | - |
| CHEMBL1372691 | — | IC50 | > | 29916.0 | nM | - |
| CHEMBL1490948 | — | IC50 | > | 29910.0 | nM | - |
| CHEMBL1896865 | — | IC50 | > | 29908.0 | nM | - |
| CHEMBL3189778 | — | IC50 | > | 29909.0 | nM | - |
| CHEMBL1525419 | — | IC50 | > | 29881.0 | nM | - |
| CHEMBL1877432 | — | IC50 | > | 29908.0 | nM | - |
| CHEMBL1362116 | — | IC50 | > | 29908.0 | nM | - |
| CHEMBL3208641 | — | IC50 | > | 29905.0 | nM | - |
| CHEMBL1593829 | — | IC50 | > | 29910.0 | nM | - |
| CHEMBL3191107 | — | IC50 | > | 29910.0 | nM | - |
| CHEMBL1476854 | — | IC50 | > | 29907.0 | nM | - |
| CHEMBL1315467 | — | IC50 | > | 29910.0 | nM | - |
| CHEMBL1704306 | — | IC50 | > | 29902.0 | nM | - |
| CHEMBL1402878 | — | IC50 | > | 9972.0 | nM | - |
| CHEMBL3190072 | — | IC50 | > | 29910.0 | nM | - |
| CHEMBL1999268 | — | IC50 | > | 29888.0 | nM | - |
| CHEMBL1603300 | — | IC50 | > | 29909.0 | nM | - |
| CHEMBL1564914 | — | IC50 | > | 29905.0 | nM | - |
| CHEMBL1375903 | — | IC50 | > | 29908.0 | nM | - |
| CHEMBL1521368 | — | IC50 | > | 29906.0 | nM | - |