Assay Detail
Functional
CHEMBL2354292
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PubChem BioAssay. Luminescence-based cell-based high throughput dose response assay for inhibitors of the orphan nuclear receptor subfamily 0, group B, member 1 (DAX1; NR0B1): repression of SF-1 (NR5A1) activated StAR promoter by full-length DAX-1. (Class of assay: confirmatory)
249
Total Activities
249
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Nuclear receptor subfamily 0 group B member 1 (CHEMBL1795094) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 249 | 5.52 | 6.87 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL19980 | BREFELDIN A | — | 1 | 6.87 |
| CHEMBL434976 | — | — | 1 | 6.67 |
| CHEMBL1706279 | — | — | 1 | 6.61 |
| CHEMBL1734496 | — | — | 1 | 6.41 |
| CHEMBL98 | VORINOSTAT | 4.0 | 1 | 6.13 |
| CHEMBL1524921 | — | — | 1 | 5.84 |
| CHEMBL52606 | COLFORSIN | 2.0 | 1 | 5.76 |
| CHEMBL3199267 | — | — | 1 | 5.68 |
| CHEMBL61 | PODOFILOX | 4.0 | 1 | 5.67 |
| CHEMBL1707859 | — | — | 1 | 5.57 |
| CHEMBL1506679 | — | — | 1 | 5.10 |
| CHEMBL1718241 | — | — | 1 | 4.99 |
| CHEMBL2361294 | — | — | 1 | 4.85 |
| CHEMBL1736008 | — | — | 1 | 4.80 |
| CHEMBL1567097 | — | — | 1 | 4.76 |
| CHEMBL1322487 | — | — | 1 | 4.61 |
| CHEMBL1324620 | — | — | 1 | 4.50 |
| CHEMBL77552 | CENTAUREIDIN | — | 1 | 4.46 |
| CHEMBL1464327 | — | — | 1 | - |
| CHEMBL1575124 | — | — | 1 | - |
| CHEMBL1599090 | — | — | 1 | - |
| CHEMBL1454840 | — | — | 1 | - |
| CHEMBL1386036 | — | — | 1 | - |
| CHEMBL1358011 | — | — | 1 | - |
| CHEMBL1575293 | — | — | 1 | - |
| CHEMBL1526661 | — | — | 1 | - |
| CHEMBL277648 | — | — | 1 | - |
| CHEMBL1565955 | — | — | 1 | - |
| CHEMBL107 | COLCHICINE | 4.0 | 1 | - |
| CHEMBL1447068 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL19980 | BREFELDIN A | IC50 | = | 134.26 | nM | 6.87 |
| CHEMBL434976 | — | IC50 | = | 212.03 | nM | 6.67 |
| CHEMBL1706279 | — | IC50 | = | 244.15 | nM | 6.61 |
| CHEMBL1734496 | — | IC50 | = | 386.05 | nM | 6.41 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 747.17 | nM | 6.13 |
| CHEMBL1524921 | — | IC50 | = | 1432.0 | nM | 5.84 |
| CHEMBL52606 | COLFORSIN | IC50 | = | 1729.0 | nM | 5.76 |
| CHEMBL3199267 | — | IC50 | = | 2094.0 | nM | 5.68 |
| CHEMBL61 | PODOFILOX | IC50 | = | 2145.0 | nM | 5.67 |
| CHEMBL1707859 | — | IC50 | = | 2715.0 | nM | 5.57 |
| CHEMBL1506679 | — | IC50 | = | 7904.0 | nM | 5.10 |
| CHEMBL1718241 | — | IC50 | = | 10314.0 | nM | 4.99 |
| CHEMBL2361294 | — | IC50 | = | 14029.0 | nM | 4.85 |
| CHEMBL1736008 | — | IC50 | = | 15803.0 | nM | 4.80 |
| CHEMBL1567097 | — | IC50 | = | 17554.0 | nM | 4.76 |
| CHEMBL1322487 | — | IC50 | = | 24722.0 | nM | 4.61 |
| CHEMBL1324620 | — | IC50 | = | 31745.0 | nM | 4.50 |
| CHEMBL77552 | CENTAUREIDIN | IC50 | = | 34985.0 | nM | 4.46 |
| CHEMBL1349455 | — | IC50 | > | 67527.0 | nM | - |
| CHEMBL1321427 | — | IC50 | > | 67574.0 | nM | - |
| CHEMBL1318263 | — | IC50 | > | 833.72 | nM | - |
| CHEMBL1569621 | — | IC50 | > | 833.93 | nM | - |
| CHEMBL1467943 | — | IC50 | > | 67541.0 | nM | - |
| CHEMBL1428850 | — | IC50 | > | 833.59 | nM | - |
| CHEMBL1321603 | — | IC50 | > | 67588.0 | nM | - |
| CHEMBL1422450 | — | IC50 | > | 67520.0 | nM | - |
| CHEMBL1727807 | — | IC50 | > | 67466.0 | nM | - |
| CHEMBL1500581 | — | IC50 | > | 67554.0 | nM | - |
| CHEMBL1433494 | — | IC50 | > | 67539.0 | nM | - |
| CHEMBL1390171 | — | IC50 | > | 67568.0 | nM | - |
| CHEMBL1484968 | — | IC50 | > | 2499.0 | nM | - |
| CHEMBL1354361 | — | IC50 | > | 67516.0 | nM | - |
| CHEMBL2142604 | — | IC50 | > | 67554.0 | nM | - |
| CHEMBL1597334 | — | IC50 | > | 67490.0 | nM | - |
| CHEMBL320802 | — | IC50 | > | 67539.0 | nM | - |
| CHEMBL1552047 | — | IC50 | > | 67533.0 | nM | - |
| CHEMBL1336651 | — | IC50 | > | 67581.0 | nM | - |
| CHEMBL1310496 | — | IC50 | > | 2502.0 | nM | - |
| CHEMBL1563383 | — | IC50 | > | 277.73 | nM | - |
| CHEMBL1383700 | — | IC50 | > | 67539.0 | nM | - |
| CHEMBL1310773 | — | IC50 | > | 67588.0 | nM | - |
| CHEMBL1453121 | — | IC50 | > | 67547.0 | nM | - |
| CHEMBL1343831 | — | IC50 | > | 67547.0 | nM | - |
| CHEMBL1878855 | — | IC50 | > | 67488.0 | nM | - |
| CHEMBL2143334 | — | IC50 | > | 67574.0 | nM | - |
| CHEMBL1531903 | — | IC50 | > | 67602.0 | nM | - |
| CHEMBL2143132 | — | IC50 | > | 67568.0 | nM | - |
| CHEMBL9514 | NOCODAZOLE | IC50 | > | 833.38 | nM | - |
| CHEMBL1375043 | — | IC50 | > | 67479.0 | nM | - |
| CHEMBL1532083 | — | IC50 | > | 67574.0 | nM | - |