Assay Detail
Functional
CHEMBL2363153
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SANGER: Inhibition of human CTV-1 cell growth in a cell viability assay.
126
Total Activities
125
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CTV-1 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 126 | 5.98 | 10.50 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL213100 | — | — | 1 | 10.50 |
| CHEMBL5416410 | DASATINIB | 4.0 | 1 | 10.39 |
| CHEMBL197603 | — | — | 1 | 10.31 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 9.04 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.85 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 8.55 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.47 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.30 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.29 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 8.28 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 8.28 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 7.85 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 7.83 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.79 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 7.73 |
| CHEMBL514499 | GW843682X | — | 1 | 7.52 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.48 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 7.41 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.39 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 7.26 |
| CHEMBL217092 | SARACATINIB | 3.0 | 1 | 7.21 |
| CHEMBL300389 | — | — | 1 | 7.18 |
| CHEMBL1256459 | TORIN1 | — | 1 | 7.18 |
| CHEMBL512504 | — | — | 1 | 7.14 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 7.12 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 7.11 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 7.07 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 7.06 |
| CHEMBL288441 | BOSUTINIB | 4.0 | 1 | 6.79 |
| CHEMBL1090090 | VX-702 | 2.0 | 1 | 6.74 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL213100 | — | IC50 | = | 0.03182 | nM | 10.50 |
| CHEMBL5416410 | DASATINIB | IC50 | = | 0.04036 | nM | 10.39 |
| CHEMBL197603 | — | IC50 | = | 0.04902 | nM | 10.31 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 0.9054 | nM | 9.04 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 1.405 | nM | 8.85 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 2.799 | nM | 8.55 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 3.371 | nM | 8.47 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 5.011 | nM | 8.30 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 5.16 | nM | 8.29 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 5.196 | nM | 8.28 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 5.206 | nM | 8.28 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 14.14 | nM | 7.85 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 14.78 | nM | 7.83 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 16.07 | nM | 7.79 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 18.67 | nM | 7.73 |
| CHEMBL514499 | GW843682X | IC50 | = | 30.39 | nM | 7.52 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 32.82 | nM | 7.48 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 38.96 | nM | 7.41 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 41.16 | nM | 7.39 |
| CHEMBL513909 | BI-2536 | IC50 | = | 55.02 | nM | 7.26 |
| CHEMBL217092 | SARACATINIB | IC50 | = | 61.43 | nM | 7.21 |
| CHEMBL300389 | — | IC50 | = | 66.0 | nM | 7.18 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 65.48 | nM | 7.18 |
| CHEMBL512504 | — | IC50 | = | 73.03 | nM | 7.14 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 75.17 | nM | 7.12 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 77.1 | nM | 7.11 |
| CHEMBL803 | CYTARABINE | IC50 | = | 84.74 | nM | 7.07 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 86.41 | nM | 7.06 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 163.98 | nM | 6.79 |
| CHEMBL1090090 | VX-702 | IC50 | = | 183.89 | nM | 6.74 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 188.92 | nM | 6.72 |
| CHEMBL379300 | A-443654 | IC50 | = | 323.24 | nM | 6.49 |
| CHEMBL585951 | — | IC50 | = | 405.22 | nM | 6.39 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 409.69 | nM | 6.39 |
| CHEMBL573107 | — | IC50 | = | 478.72 | nM | 6.32 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 526.69 | nM | 6.28 |
| CHEMBL509032 | TAE-684 | IC50 | = | 556.24 | nM | 6.25 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 581.56 | nM | 6.24 |
| CHEMBL572878 | TOZASERTIB | IC50 | = | 587.73 | nM | 6.23 |
| CHEMBL601719 | CRIZOTINIB | IC50 | = | 596.48 | nM | 6.22 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 643.92 | nM | 6.19 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 744.9 | nM | 6.13 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | IC50 | = | 787.8 | nM | 6.10 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 854.73 | nM | 6.07 |
| CHEMBL38 | TRETINOIN | IC50 | = | 962.82 | nM | 6.02 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 1046.56 | nM | 5.98 |
| CHEMBL2144069 | — | IC50 | = | 1200.65 | nM | 5.92 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 1274.25 | nM | 5.89 |
| CHEMBL939 | GEFITINIB | IC50 | = | 1308.0 | nM | 5.88 |
| CHEMBL1190711 | — | IC50 | = | 1496.31 | nM | 5.83 |