Assay Detail
Functional
CHEMBL2363229
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SANGER: Inhibition of human EW-7 cell growth in a cell viability assay.
47
Total Activities
46
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | EW-7 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 47 | 6.00 | 8.76 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 8.76 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.65 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 8.20 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 8.12 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 7.92 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.78 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.51 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 7.21 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 6.90 |
| CHEMBL217354 | — | — | 1 | 6.78 |
| CHEMBL1091644 | LINSITINIB | 3.0 | 1 | 6.72 |
| CHEMBL585951 | — | — | 1 | 6.25 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.17 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.11 |
| CHEMBL2165191 | AZD-6482 | 2.0 | 2 | 6.06 |
| CHEMBL9470 | SHIKONIN | — | 1 | 5.89 |
| CHEMBL1190711 | — | — | 1 | 5.70 |
| CHEMBL2137530 | SERDEMETAN | 2.0 | 1 | 5.63 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 5.51 |
| CHEMBL1173055 | RUCAPARIB | 4.0 | 1 | 5.45 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 5.43 |
| CHEMBL1186585 | — | — | 1 | 5.08 |
| CHEMBL591429 | PAC-1 | 1.0 | 1 | 4.99 |
| CHEMBL1084546 | PF-00562271 | 1.0 | 1 | 4.70 |
| CHEMBL2134202 | — | — | 1 | 4.68 |
| CHEMBL221137 | EMBELIN | — | 1 | 4.63 |
| CHEMBL258844 | — | — | 1 | 4.45 |
| CHEMBL228043 | — | — | 1 | 4.36 |
| CHEMBL191384 | — | — | 1 | 4.28 |
| CHEMBL135561 | — | — | 1 | 4.20 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 1.754 | nM | 8.76 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 2.245 | nM | 8.65 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 6.345 | nM | 8.20 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 7.54 | nM | 8.12 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 12.14 | nM | 7.92 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 16.7 | nM | 7.78 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 30.63 | nM | 7.51 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 61.01 | nM | 7.21 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 125.06 | nM | 6.90 |
| CHEMBL217354 | — | IC50 | = | 166.87 | nM | 6.78 |
| CHEMBL1091644 | LINSITINIB | IC50 | = | 188.81 | nM | 6.72 |
| CHEMBL585951 | — | IC50 | = | 561.5 | nM | 6.25 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 681.95 | nM | 6.17 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 781.09 | nM | 6.11 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 863.56 | nM | 6.06 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 1290.91 | nM | 5.89 |
| CHEMBL1190711 | — | IC50 | = | 1977.91 | nM | 5.70 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 2326.95 | nM | 5.63 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 3058.66 | nM | 5.51 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 3106.0 | nM | 5.51 |
| CHEMBL1173055 | RUCAPARIB | IC50 | = | 3570.69 | nM | 5.45 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 3676.93 | nM | 5.43 |
| CHEMBL1186585 | — | IC50 | = | 8295.32 | nM | 5.08 |
| CHEMBL591429 | PAC-1 | IC50 | = | 10228.33 | nM | 4.99 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 20162.83 | nM | 4.70 |
| CHEMBL2134202 | — | IC50 | = | 20858.76 | nM | 4.68 |
| CHEMBL221137 | EMBELIN | IC50 | = | 23177.25 | nM | 4.63 |
| CHEMBL258844 | — | IC50 | = | 35409.67 | nM | 4.45 |
| CHEMBL228043 | — | IC50 | = | 43985.37 | nM | 4.36 |
| CHEMBL191384 | — | IC50 | = | 53050.17 | nM | 4.28 |
| CHEMBL135561 | — | IC50 | = | 63606.9 | nM | 4.20 |
| CHEMBL512504 | — | IC50 | = | 66968.28 | nM | 4.17 |
| CHEMBL409 | BICALUTAMIDE | IC50 | = | 70737.58 | nM | 4.15 |
| CHEMBL472940 | — | IC50 | = | 302021.14 | nM | - |
| CHEMBL558642 | GSK-650394 | IC50 | = | 471144.57 | nM | - |
| CHEMBL2363137 | — | IC50 | = | 144054.69 | nM | - |
| CHEMBL92309 | — | IC50 | = | 729063.62 | nM | - |
| CHEMBL1023 | BEXAROTENE | IC50 | = | 495778.87 | nM | - |
| CHEMBL412142 | LADUVIGLUSIB | IC50 | = | 285232.32 | nM | - |
| CHEMBL259181 | — | IC50 | = | 182935.02 | nM | - |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 164109.35 | nM | - |
| CHEMBL477772 | PAZOPANIB | IC50 | = | 677505.72 | nM | - |
| CHEMBL888 | GEMCITABINE | IC50 | = | 0.002578 | nM | - |
| CHEMBL255342 | — | IC50 | = | 264468.72 | nM | - |
| CHEMBL399530 | — | IC50 | = | 132535.03 | nM | - |
| CHEMBL472004 | — | IC50 | = | 2115583.63 | nM | - |
| CHEMBL1090771 | AVAGACESTAT | IC50 | = | 158247.46 | nM | - |