Assay Detail
Functional
CHEMBL2363233
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SANGER: Inhibition of human G-361 cell growth in a cell viability assay.
79
Total Activities
78
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | G-361 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 79 | 5.92 | 9.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 9.15 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 8.91 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.45 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.97 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 7.86 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 7.68 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.57 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.56 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.55 |
| CHEMBL512504 | — | — | 1 | 7.05 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 7.05 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 6.91 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.91 |
| CHEMBL217354 | — | — | 1 | 6.90 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 6.84 |
| CHEMBL176544 | — | — | 1 | 6.68 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.68 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.66 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.64 |
| CHEMBL585951 | — | — | 1 | 6.58 |
| CHEMBL1289926 | AXITINIB | 4.0 | 1 | 6.49 |
| CHEMBL1230020 | PLX-4720 | — | 1 | 6.46 |
| CHEMBL105442 | CI-1040 | 2.0 | 1 | 6.43 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.41 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.33 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 6.09 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 6.08 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 5.99 |
| CHEMBL289228 | TIPIFARNIB | 3.0 | 1 | 5.94 |
| CHEMBL591429 | PAC-1 | 1.0 | 1 | 5.92 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | IC50 | = | 0.7013 | nM | 9.15 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 1.24 | nM | 8.91 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 3.525 | nM | 8.45 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 10.67 | nM | 7.97 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 13.93 | nM | 7.86 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 21.07 | nM | 7.68 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 26.77 | nM | 7.57 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 27.54 | nM | 7.56 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 27.88 | nM | 7.55 |
| CHEMBL512504 | — | IC50 | = | 88.15 | nM | 7.05 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 88.31 | nM | 7.05 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 123.24 | nM | 6.91 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 123.93 | nM | 6.91 |
| CHEMBL217354 | — | IC50 | = | 124.95 | nM | 6.90 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 145.66 | nM | 6.84 |
| CHEMBL176544 | — | IC50 | = | 210.6 | nM | 6.68 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 208.53 | nM | 6.68 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 221.08 | nM | 6.66 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 226.82 | nM | 6.64 |
| CHEMBL585951 | — | IC50 | = | 265.8 | nM | 6.58 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 323.25 | nM | 6.49 |
| CHEMBL1230020 | PLX-4720 | IC50 | = | 346.37 | nM | 6.46 |
| CHEMBL105442 | CI-1040 | IC50 | = | 367.95 | nM | 6.43 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 387.12 | nM | 6.41 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 473.21 | nM | 6.33 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 818.97 | nM | 6.09 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 833.87 | nM | 6.08 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 1035.15 | nM | 5.99 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 1138.94 | nM | 5.94 |
| CHEMBL591429 | PAC-1 | IC50 | = | 1187.64 | nM | 5.92 |
| CHEMBL1090090 | VX-702 | IC50 | = | 1495.19 | nM | 5.83 |
| CHEMBL2363137 | — | IC50 | = | 1769.39 | nM | 5.75 |
| CHEMBL259181 | — | IC50 | = | 2055.56 | nM | 5.69 |
| CHEMBL573107 | — | IC50 | = | 2122.1 | nM | 5.67 |
| CHEMBL188678 | — | IC50 | = | 2216.8 | nM | 5.65 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 2544.45 | nM | 5.59 |
| CHEMBL477772 | PAZOPANIB | IC50 | = | 3040.82 | nM | 5.52 |
| CHEMBL558642 | GSK-650394 | IC50 | = | 3717.45 | nM | 5.43 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 3899.94 | nM | 5.41 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 4090.6 | nM | 5.39 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 4123.67 | nM | 5.38 |
| CHEMBL1190711 | — | IC50 | = | 4297.26 | nM | 5.37 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 5010.03 | nM | 5.30 |
| CHEMBL221137 | EMBELIN | IC50 | = | 5897.66 | nM | 5.23 |
| CHEMBL412142 | LADUVIGLUSIB | IC50 | = | 7465.61 | nM | 5.13 |
| CHEMBL102714 | SB-216763 | IC50 | = | 10179.76 | nM | 4.99 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 10674.91 | nM | 4.97 |
| CHEMBL939 | GEFITINIB | IC50 | = | 12912.89 | nM | 4.89 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 13666.4 | nM | 4.86 |
| CHEMBL409 | BICALUTAMIDE | IC50 | = | 17825.96 | nM | 4.75 |