Assay Detail
Functional
CHEMBL2363239
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SANGER: Inhibition of human GCIY cell growth in a cell viability assay.
139
Total Activities
137
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | GCIY |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 139 | 5.61 | 8.79 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 8.79 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.18 |
| CHEMBL1256459 | TORIN1 | — | 1 | 8.00 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.69 |
| CHEMBL217354 | — | — | 1 | 7.68 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 7.60 |
| CHEMBL9470 | SHIKONIN | — | 1 | 7.44 |
| CHEMBL514499 | GW843682X | — | 1 | 7.32 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 7.30 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.29 |
| CHEMBL413 | SIROLIMUS | 4.0 | 1 | 7.27 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.27 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.24 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 7.18 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 7.03 |
| CHEMBL5416410 | DASATINIB | 4.0 | 1 | 7.01 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 6.95 |
| CHEMBL585951 | — | — | 1 | 6.89 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 6.83 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.74 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 6.60 |
| CHEMBL379300 | A-443654 | — | 1 | 6.58 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.54 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.51 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 6.48 |
| CHEMBL401930 | — | — | 1 | 6.39 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.39 |
| CHEMBL521851 | PICTILISIB | 2.0 | 1 | 6.36 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.34 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 6.32 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 1.625 | nM | 8.79 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 6.592 | nM | 8.18 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 10.07 | nM | 8.00 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 20.55 | nM | 7.69 |
| CHEMBL217354 | — | IC50 | = | 20.83 | nM | 7.68 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 25.02 | nM | 7.60 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 35.98 | nM | 7.44 |
| CHEMBL514499 | GW843682X | IC50 | = | 47.98 | nM | 7.32 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 49.73 | nM | 7.30 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 50.67 | nM | 7.29 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 53.46 | nM | 7.27 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 53.46 | nM | 7.27 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 57.88 | nM | 7.24 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 66.15 | nM | 7.18 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 92.69 | nM | 7.03 |
| CHEMBL5416410 | DASATINIB | IC50 | = | 96.56 | nM | 7.01 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 111.82 | nM | 6.95 |
| CHEMBL585951 | — | IC50 | = | 129.43 | nM | 6.89 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 149.01 | nM | 6.83 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 183.37 | nM | 6.74 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 253.75 | nM | 6.60 |
| CHEMBL379300 | A-443654 | IC50 | = | 261.31 | nM | 6.58 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 286.92 | nM | 6.54 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 310.02 | nM | 6.51 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 328.74 | nM | 6.48 |
| CHEMBL401930 | — | IC50 | = | 404.28 | nM | 6.39 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 410.99 | nM | 6.39 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 433.8 | nM | 6.36 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 457.54 | nM | 6.34 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 484.53 | nM | 6.32 |
| CHEMBL513909 | BI-2536 | IC50 | = | 703.63 | nM | 6.15 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 725.12 | nM | 6.14 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 918.43 | nM | 6.04 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 925.49 | nM | 6.03 |
| CHEMBL509032 | TAE-684 | IC50 | = | 955.26 | nM | 6.02 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 1081.04 | nM | 5.97 |
| CHEMBL300389 | — | IC50 | = | 1136.08 | nM | 5.95 |
| CHEMBL3349342 | — | IC50 | = | 1181.23 | nM | 5.93 |
| CHEMBL213100 | — | IC50 | = | 1230.1 | nM | 5.91 |
| CHEMBL939 | GEFITINIB | IC50 | = | 1301.32 | nM | 5.89 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 1390.51 | nM | 5.86 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | IC50 | = | 1818.63 | nM | 5.74 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 2199.28 | nM | 5.66 |
| CHEMBL803 | CYTARABINE | IC50 | = | 2802.34 | nM | 5.55 |
| CHEMBL217092 | SARACATINIB | IC50 | = | 2870.05 | nM | 5.54 |
| CHEMBL2363137 | — | IC50 | = | 2944.11 | nM | 5.53 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 3204.91 | nM | 5.49 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 3921.37 | nM | 5.41 |
| CHEMBL197603 | — | IC50 | = | 4034.66 | nM | 5.39 |
| CHEMBL553 | ERLOTINIB | IC50 | = | 4635.32 | nM | 5.33 |