Assay Detail
Functional
CHEMBL2363308
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SANGER: Inhibition of human IGR-1 cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | IGR-1 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.76 | 9.06 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 9.06 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.72 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.68 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 8.22 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.19 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.98 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 7.84 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.69 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.47 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 7.36 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.34 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 6.82 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.81 |
| CHEMBL585951 | — | — | 1 | 6.78 |
| CHEMBL217354 | — | — | 1 | 6.52 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.49 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 6.46 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.41 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 6.12 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.10 |
| CHEMBL1090771 | AVAGACESTAT | 2.0 | 1 | 5.98 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 5.97 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 5.83 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 5.80 |
| CHEMBL289228 | TIPIFARNIB | 3.0 | 1 | 5.79 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 5.75 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 5.75 |
| CHEMBL2363137 | — | — | 1 | 5.70 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 5.63 |
| CHEMBL443684 | NAVITOCLAX | 3.0 | 1 | 5.58 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | IC50 | = | 0.8634 | nM | 9.06 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 1.903 | nM | 8.72 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 2.076 | nM | 8.68 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 6.012 | nM | 8.22 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 6.414 | nM | 8.19 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 10.51 | nM | 7.98 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 14.42 | nM | 7.84 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 20.5 | nM | 7.69 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 33.88 | nM | 7.47 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 43.71 | nM | 7.36 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 46.13 | nM | 7.34 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 151.26 | nM | 6.82 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 153.98 | nM | 6.81 |
| CHEMBL585951 | — | IC50 | = | 164.41 | nM | 6.78 |
| CHEMBL217354 | — | IC50 | = | 300.61 | nM | 6.52 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 321.6 | nM | 6.49 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 345.07 | nM | 6.46 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 393.69 | nM | 6.41 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 767.16 | nM | 6.12 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 790.43 | nM | 6.10 |
| CHEMBL1090771 | AVAGACESTAT | IC50 | = | 1047.78 | nM | 5.98 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 1063.61 | nM | 5.97 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 1492.37 | nM | 5.83 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 1591.12 | nM | 5.80 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 1624.6 | nM | 5.79 |
| CHEMBL803 | CYTARABINE | IC50 | = | 1782.79 | nM | 5.75 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 1756.71 | nM | 5.75 |
| CHEMBL2363137 | — | IC50 | = | 2011.32 | nM | 5.70 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 2346.33 | nM | 5.63 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 2620.35 | nM | 5.58 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 2738.74 | nM | 5.56 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 2839.87 | nM | 5.55 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 3120.28 | nM | 5.51 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 3742.48 | nM | 5.43 |
| CHEMBL573107 | — | IC50 | = | 4102.74 | nM | 5.39 |
| CHEMBL558642 | GSK-650394 | IC50 | = | 4233.0 | nM | 5.37 |
| CHEMBL191384 | — | IC50 | = | 4678.66 | nM | 5.33 |
| CHEMBL3349342 | — | IC50 | = | 5009.78 | nM | 5.30 |
| CHEMBL221137 | EMBELIN | IC50 | = | 5383.63 | nM | 5.27 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 5868.94 | nM | 5.23 |
| CHEMBL577784 | BX-795 | IC50 | = | 5889.78 | nM | 5.23 |
| CHEMBL399530 | — | IC50 | = | 5993.94 | nM | 5.22 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 6452.14 | nM | 5.19 |
| CHEMBL1190711 | — | IC50 | = | 6537.71 | nM | 5.18 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 6978.26 | nM | 5.16 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 8180.51 | nM | 5.09 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 8430.23 | nM | 5.07 |
| CHEMBL259181 | — | IC50 | = | 11385.65 | nM | 4.94 |
| CHEMBL191334 | NUTLIN-3 | IC50 | = | 14034.7 | nM | 4.85 |
| CHEMBL1186585 | — | IC50 | = | 16632.11 | nM | 4.78 |