Assay Detail
Functional
CHEMBL2363436
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SANGER: Inhibition of human MOLT-13 cell growth in a cell viability assay.
60
Total Activities
60
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | MOLT-13 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 60 | 5.55 | 8.75 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 8.75 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.25 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 7.96 |
| CHEMBL514499 | GW843682X | — | 1 | 7.92 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 7.79 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 7.37 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 6.95 |
| CHEMBL1090090 | VX-702 | 2.0 | 1 | 6.80 |
| CHEMBL1173655 | AFATINIB | 4.0 | 1 | 6.62 |
| CHEMBL1256459 | TORIN1 | — | 1 | 6.52 |
| CHEMBL27759 | ENTINOSTAT | 3.0 | 1 | 6.47 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.39 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.33 |
| CHEMBL443684 | NAVITOCLAX | 3.0 | 1 | 6.33 |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | 6.29 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.18 |
| CHEMBL98 | VORINOSTAT | 4.0 | 1 | 6.13 |
| CHEMBL189963 | PALBOCICLIB | 4.0 | 1 | 5.99 |
| CHEMBL38 | TRETINOIN | 4.0 | 1 | 5.94 |
| CHEMBL202721 | — | — | 1 | 5.80 |
| CHEMBL573107 | — | — | 1 | 5.40 |
| CHEMBL1614701 | SELUMETINIB | 4.0 | 1 | 5.39 |
| CHEMBL220241 | GSK-269962A | — | 1 | 5.35 |
| CHEMBL105442 | CI-1040 | 2.0 | 1 | 5.29 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 5.25 |
| CHEMBL2144069 | — | — | 1 | 5.23 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 5.07 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 4.77 |
| CHEMBL1289926 | AXITINIB | 4.0 | 1 | 4.71 |
| CHEMBL3349342 | — | — | 1 | 4.67 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 1.787 | nM | 8.75 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 5.603 | nM | 8.25 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 10.86 | nM | 7.96 |
| CHEMBL514499 | GW843682X | IC50 | = | 12.09 | nM | 7.92 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 16.37 | nM | 7.79 |
| CHEMBL513909 | BI-2536 | IC50 | = | 42.38 | nM | 7.37 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 113.44 | nM | 6.95 |
| CHEMBL1090090 | VX-702 | IC50 | = | 159.81 | nM | 6.80 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 239.75 | nM | 6.62 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 301.83 | nM | 6.52 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 338.1 | nM | 6.47 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 408.52 | nM | 6.39 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 462.94 | nM | 6.33 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 466.13 | nM | 6.33 |
| CHEMBL939 | GEFITINIB | IC50 | = | 514.82 | nM | 6.29 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 665.37 | nM | 6.18 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 738.98 | nM | 6.13 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 1014.21 | nM | 5.99 |
| CHEMBL38 | TRETINOIN | IC50 | = | 1145.0 | nM | 5.94 |
| CHEMBL202721 | — | IC50 | = | 1567.06 | nM | 5.80 |
| CHEMBL573107 | — | IC50 | = | 3968.56 | nM | 5.40 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 4034.19 | nM | 5.39 |
| CHEMBL220241 | GSK-269962A | IC50 | = | 4436.53 | nM | 5.35 |
| CHEMBL105442 | CI-1040 | IC50 | = | 5067.76 | nM | 5.29 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 5554.3 | nM | 5.25 |
| CHEMBL2144069 | — | IC50 | = | 5828.67 | nM | 5.23 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 8595.11 | nM | 5.07 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 16918.79 | nM | 4.77 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 19454.57 | nM | 4.71 |
| CHEMBL3349342 | — | IC50 | = | 21270.03 | nM | 4.67 |
| CHEMBL521686 | OLAPARIB | IC50 | = | 25533.13 | nM | 4.59 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 25674.36 | nM | 4.59 |
| CHEMBL209148 | — | IC50 | = | 25997.57 | nM | 4.58 |
| CHEMBL450786 | PHA-665752 | IC50 | = | 27184.75 | nM | 4.57 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 27351.57 | nM | 4.56 |
| CHEMBL506871 | VELIPARIB | IC50 | = | 29381.43 | nM | 4.53 |
| CHEMBL477989 | SB590885 | IC50 | = | 30867.88 | nM | 4.51 |
| CHEMBL401930 | — | IC50 | = | 35079.43 | nM | 4.46 |
| CHEMBL180127 | SALUBRINAL | IC50 | = | 35662.44 | nM | 4.45 |
| CHEMBL189584 | PD-173074 | IC50 | = | 39250.18 | nM | 4.41 |
| CHEMBL803 | CYTARABINE | IC50 | = | 58554.21 | nM | 4.23 |
| CHEMBL1230020 | PLX-4720 | IC50 | = | 58566.63 | nM | 4.23 |
| CHEMBL255863 | NILOTINIB | IC50 | = | 58574.47 | nM | 4.23 |
| CHEMBL36 | PYRIMETHAMINE | IC50 | = | 66334.43 | nM | 4.18 |
| CHEMBL191334 | NUTLIN-3 | IC50 | = | 85239.42 | nM | 4.07 |
| CHEMBL848 | LENALIDOMIDE | IC50 | = | 87224.3 | nM | 4.06 |
| CHEMBL1336 | SORAFENIB | IC50 | = | 90128.37 | nM | 4.04 |
| CHEMBL379975 | — | IC50 | = | 97527.17 | nM | 4.01 |
| CHEMBL217092 | SARACATINIB | IC50 | = | 578017.99 | nM | - |
| CHEMBL176544 | — | IC50 | = | 144647.97 | nM | - |