Assay Detail
Functional
CHEMBL2363444
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SANGER: Inhibition of human MV-4-11 cell growth in a cell viability assay.
129
Total Activities
128
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | MV-4-11 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 129 | 6.33 | 10.02 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 10.02 |
| CHEMBL535 | SUNITINIB | 4.0 | 1 | 9.56 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 9.48 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 9.37 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 9.25 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 9.15 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.77 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 8.76 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.76 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 8.74 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.55 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 8.32 |
| CHEMBL1190711 | — | — | 1 | 8.13 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 8.00 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 8.00 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.98 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.96 |
| CHEMBL443684 | NAVITOCLAX | 3.0 | 1 | 7.80 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.75 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.72 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 7.71 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 7.70 |
| CHEMBL38 | TRETINOIN | 4.0 | 1 | 7.68 |
| CHEMBL512504 | — | — | 1 | 7.64 |
| CHEMBL514499 | GW843682X | — | 1 | 7.59 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.54 |
| CHEMBL577784 | BX-795 | — | 1 | 7.43 |
| CHEMBL300389 | — | — | 1 | 7.37 |
| CHEMBL379300 | A-443654 | — | 1 | 7.24 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 7.17 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1171837 | PONATINIB | IC50 | = | 0.09555 | nM | 10.02 |
| CHEMBL535 | SUNITINIB | IC50 | = | 0.2722 | nM | 9.56 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 0.3337 | nM | 9.48 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 0.4245 | nM | 9.37 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 0.5585 | nM | 9.25 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 0.7058 | nM | 9.15 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 1.696 | nM | 8.77 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 1.744 | nM | 8.76 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 1.732 | nM | 8.76 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 1.817 | nM | 8.74 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 2.805 | nM | 8.55 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 4.747 | nM | 8.32 |
| CHEMBL1190711 | — | IC50 | = | 7.394 | nM | 8.13 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 10.03 | nM | 8.00 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 9.908 | nM | 8.00 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 10.39 | nM | 7.98 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 10.98 | nM | 7.96 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 15.86 | nM | 7.80 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 18.0 | nM | 7.75 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 18.88 | nM | 7.72 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 19.35 | nM | 7.71 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 19.83 | nM | 7.70 |
| CHEMBL38 | TRETINOIN | IC50 | = | 20.99 | nM | 7.68 |
| CHEMBL512504 | — | IC50 | = | 22.74 | nM | 7.64 |
| CHEMBL514499 | GW843682X | IC50 | = | 25.89 | nM | 7.59 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 28.7 | nM | 7.54 |
| CHEMBL577784 | BX-795 | IC50 | = | 36.8 | nM | 7.43 |
| CHEMBL300389 | — | IC50 | = | 43.1 | nM | 7.37 |
| CHEMBL379300 | A-443654 | IC50 | = | 57.74 | nM | 7.24 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 68.03 | nM | 7.17 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 69.95 | nM | 7.16 |
| CHEMBL572878 | TOZASERTIB | IC50 | = | 77.82 | nM | 7.11 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 83.73 | nM | 7.08 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 94.73 | nM | 7.02 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 103.47 | nM | 6.99 |
| CHEMBL220241 | GSK-269962A | IC50 | = | 139.15 | nM | 6.86 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 151.21 | nM | 6.82 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 162.64 | nM | 6.79 |
| CHEMBL558642 | GSK-650394 | IC50 | = | 164.9 | nM | 6.78 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 179.77 | nM | 6.75 |
| CHEMBL401930 | — | IC50 | = | 206.37 | nM | 6.68 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 273.63 | nM | 6.56 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 276.6 | nM | 6.56 |
| CHEMBL176544 | — | IC50 | = | 295.09 | nM | 6.53 |
| CHEMBL513909 | BI-2536 | IC50 | = | 307.88 | nM | 6.51 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | IC50 | = | 380.61 | nM | 6.42 |
| CHEMBL509032 | TAE-684 | IC50 | = | 394.46 | nM | 6.40 |
| CHEMBL1023 | BEXAROTENE | IC50 | = | 452.56 | nM | 6.34 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 513.85 | nM | 6.29 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 530.41 | nM | 6.28 |